Shipping with this method takes 3-5 days
Tolterodine LA Capsules for Overactive Bladder
Stock up and Save - Get 20% off when you buy 3 or more of any one product. Use code SAVE20 at checkout.
Coupon code cannot be combined with other offers. Sale applies to all products originating from Canada. Maximum allowable quantity equal to a 90 day supply per single order.
Price range: $77.99 through $184.99
Secure Encrypted Payments
Tolterodine LA is an extended-release capsule used to help manage overactive bladder symptoms in adults. It may reduce urgency, frequency, and urge incontinence. This page explains how it works, key safety points, dosing basics, and access options with US shipping from Canada, including choices for Tolterodine LA without insurance.
What Tolterodine LA Is and How It Works
YouDrugstore is a licensed Canadian pharmacy in Manitoba. Pharmacists review prescriptions before dispensing.
Tolterodine LA belongs to the antimuscarinic class. It relaxes bladder muscle by blocking muscarinic receptors, which can reduce involuntary contractions that cause urgency and leakage. It is the Detrol LA® generic, offering a once-daily option for sustained control. The treatment is commonly used for adults diagnosed with Overactive Bladder. For background on the condition, see What Is Overactive Bladder.
Who It’s For
This medicine is for adults with urinary urgency, frequency, and urge incontinence related to overactive bladder. People with urinary retention, gastric retention, or uncontrolled narrow-angle glaucoma should not use it. Those with significant bladder outlet obstruction, liver impairment, kidney impairment, or a history of severe constipation should discuss risks with a healthcare professional. Older adults may be more sensitive to anticholinergic effects, such as dry mouth or confusion. If you are pregnant, planning pregnancy, or breastfeeding, ask your prescriber whether this therapy is appropriate.
Dosage and Usage
The usual starting dose for the extended-release capsule is 4 mg taken once daily. Some people may use 2 mg once daily based on tolerability or other clinical factors determined by their prescriber. Swallow capsules whole with liquid. Do not crush, chew, or open the capsule contents. You can take it with or without food, ideally at the same time each day. If you have liver or kidney impairment, or take certain interacting medicines, your prescriber may choose a lower dose. When directions are unclear, follow the official label or ask a clinician.
If you are also managing other urologic conditions, you can browse related options in our Urology section.
Strengths and Forms
Extended-release capsules are commonly available in two strengths:
- 2 mg once-daily capsule
- 4 mg once-daily capsule
Availability may vary by manufacturer and time. Your prescriber will determine the appropriate strength and quantity for your prescription.
Missed Dose and Timing
If you miss a dose, take it when you remember unless it is close to your next dose. If it is almost time for the next dose, skip the missed dose. Do not take two doses at once. Keeping a simple daily reminder can help maintain a consistent schedule.
Storage and Travel Basics
Store capsules at room temperature, away from excess heat and moisture. Keep the bottle tightly closed and out of reach of children and pets. When traveling, carry your medicine in your hand luggage with the original labeled container. Pack enough for the trip and a small buffer in case of delays. If you cross time zones, take your dose based on your new local routine the next day to keep a once-daily rhythm.
Benefits
This therapy offers once-daily convenience and steady symptom control for many adults with overactive bladder. By targeting bladder muscle receptors, it may reduce urgency episodes and help increase the time between bathroom visits. Fewer interruptions can support daily activities, travel, and sleep. Consistent daily use, along with behavioral measures like fluid timing and bladder training, may improve outcomes over time.
Side Effects and Safety
- Dry mouth
- Constipation
- Headache or dizziness
- Dry eyes or blurred vision
- Indigestion or abdominal discomfort
Serious effects are less common but can include allergic reactions, trouble urinating, or severe abdominal pain. Stop the medicine and seek medical help if you experience swelling of the face, lips, tongue, or throat. Because anticholinergics can affect vision and alertness, use caution with driving or machinery until you know how you respond. If you also use insulin or sulfonylureas, monitor for dehydration from reduced fluid intake.
Drug Interactions and Cautions
Strong CYP3A4 inhibitors (for example, certain azole antifungals or macrolide antibiotics) can raise levels of this medicine. Other anticholinergics may increase side effects like dry mouth, constipation, or blurry vision. Alcohol may add to dizziness or drowsiness. Let your prescriber know about heart rhythm issues, as some medicines that affect QT interval may warrant closer evaluation. Always share a full list of your prescription drugs, OTC medicines, and supplements with your clinician.
What to Expect Over Time
Many people notice gradual improvement in urgency and frequency with regular daily use. Symptom changes can be subtle at first. Keep taking it as prescribed unless your clinician advises otherwise. If dryness is bothersome, small sips of water, sugar-free gum, or eye lubricants may help. Behavioral strategies, such as bladder training and planned bathroom breaks, can complement the medicine. Check in with your prescriber if symptoms persist, worsen, or if side effects limit use.
Compare With Alternatives
Other prescription options exist for overactive bladder. Antimuscarinics such as Solifenacin Succinate or beta-3 agonists like Myrbetriq® may be considered when appropriate. Your prescriber can compare class effects, side-effect profiles, and your medical history. For additional reading, see Myrbetriq Uses.
Pricing and Access
We aim to make access straightforward with transparent options. If you are comparing Tolterodine LA price, remember that generic formulations can help reduce cash-pay spending. We also provide guidance on comparing Detrol LA cost for patients discussing brand versus generic with a prescriber. Orders typically ship discreetly and securely. Ships from Canada to US reflects our cross-border model for eligible prescriptions. If you are looking for current promotions, visit Promotions for occasional offers.
Availability and Substitutions
Supply can vary by manufacturer and time. If a specific pack size is temporarily unavailable, your prescriber may recommend a comparable alternative in the same class or a different class based on your history and tolerability. We do not post restock dates. If you have questions about brand versus generic, ask your healthcare professional which option fits your plan and medical needs.
Patient Suitability and Cost-Saving Tips
Good candidates are adults with bothersome overactive bladder symptoms who can use an antimuscarinic safely. People with urinary retention, uncontrolled narrow-angle glaucoma, or severe gastric retention are not good candidates. To help manage spending, consider multi-month fills when your prescriber agrees, since fewer refills can lower per-fill fees. Set up refill reminders so you never miss a day. Ask about generic substitution if your prescription allows it. Some people search for a Tolterodine coupon; review any offer details carefully and discuss options with your prescriber or pharmacist. You can also explore related information in our Urinary Incontinence and Overactive Bladder pages.
Questions to Ask Your Clinician
- Is this the right antimuscarinic for my symptoms and health history?
- What signs suggest the dose or medicine should be reassessed?
- Could another bladder therapy suit me better if I have side effects?
- How should I coordinate this with my other prescriptions or eye conditions?
- What lifestyle changes could work alongside this treatment?
- When should I schedule a follow-up to review response and tolerability?
Authoritative Sources
FDA DailyMed product labeling offers the most current official information for tolterodine tartrate.
Pfizer provides brand information for Detrol LA and patient materials.
Health Canada DPD lists Canadian drug product data and monographs.
Ready to proceed? Place your order with US delivery from Canada and prompt shipping. We use temperature-controlled handling when required. Speak with your prescriber if you have clinical questions. This information is educational and not a substitute for professional medical advice.
Express Shipping - from $25.00
Prices:
- Dry-Packed Products $25.00
- Cold-Packed Products $35.00
Shipping Countries:
- United States (all contiguous states**)
- Worldwide (excludes some countries***)
Standard Shipping - $15.00
Shipping with this method takes 5-10 days
Prices:
- Dry-Packed Products $15.00
- Not available for Cold-Packed products
Shipping Countries:
- United States (all contiguous states**)
- Worldwide (excludes some countries***)
How does tolterodine extended-release differ from immediate-release?
The extended-release capsule is designed to deliver medicine steadily over 24 hours, supporting once-daily dosing. Immediate-release tablets are typically taken twice daily. Both forms use the same active ingredient, but the release profile and dosing schedule differ. If you are considering a switch, your prescriber will decide which option suits your medical history and tolerance for potential side effects like dry mouth or constipation. Always swallow the extended-release capsule whole and avoid crushing or chewing.
Can I drink alcohol while taking this medicine?
Alcohol can increase dizziness or drowsiness for some people taking antimuscarinics. If you choose to drink, do so cautiously until you understand your individual response. Avoid activities requiring alertness if you feel sedated or lightheaded. People with dehydration risk should also be mindful of fluid intake. If you have questions about specific amounts or timing with other medicines, check with your healthcare professional for personalized guidance.
What if I have glaucoma or bladder outlet obstruction?
This class can worsen certain conditions. People with uncontrolled narrow-angle glaucoma, urinary retention, or severe bladder outlet obstruction are generally not candidates. Others with milder forms may still need careful assessment and monitoring. Share your full medical history with your prescriber, including eye conditions and urinary flow issues. If you develop eye pain, changes in vision, or trouble urinating, seek medical advice promptly and stop the medicine unless told otherwise by a clinician.
How long before I notice changes in bladder symptoms?
Responses vary. Many people describe gradual improvement with daily use, though the timing and degree differ by individual factors, such as other conditions and concurrent medicines. Behavioral strategies like bladder training and timed bathroom trips may support outcomes. If symptoms persist or side effects are problematic, schedule a review with your prescriber. Do not change the dose or stop on your own without clinical advice.
Can I open the capsule if I struggle to swallow?
Do not crush, chew, or open the extended-release capsule, as that can change how the medicine is released and may increase side effects. If swallowing is difficult, ask your clinician about strategies, such as swallowing techniques, timing with water, or whether another form or alternative therapy may be appropriate. They may suggest a different medicine that better suits your needs while maintaining symptom control.
Is it safe during pregnancy or breastfeeding?
Safety data in pregnancy and breastfeeding are limited. Decisions depend on your symptoms, severity, and overall health. Discuss potential benefits and risks with your prescriber before starting or continuing the medicine. If you become pregnant while taking it, contact your healthcare professional promptly to review options. During breastfeeding, monitor the infant for anticholinergic effects, such as constipation or poor feeding, and talk with your clinician about alternatives if concerns arise.
Which medicines may interact with tolterodine?
Strong CYP3A4 inhibitors, like some azole antifungals or macrolide antibiotics, can increase blood levels and side effects. Other anticholinergics can add to dry mouth, constipation, or blurred vision. Some heart rhythm medicines may warrant extra caution. Share a complete list of prescriptions, over-the-counter products, and supplements with your prescriber and pharmacist. They can check for interactions and advise on safe timing or alternative therapies if needed.

